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Zhou Xiaoru,Li Xiao,Liao Liping,Han Jie,Huang Jing,Li Jiacheng,Tao Hongru,Fan Shijie,Chen Zhifeng,Li Qi,Chen Shijie,Ding Hong,Yang Yaxi,Zhou Bing,Jiang Hualiang,Chen Kaixian,Zhang Yuanyuan,Huang Chuanxin,Luo Cheng.P300/CBP inhibition sensitizes mantle cell lymphoma to PI3Kdelta inhibitor idelalisib[J].中国药理学报,2022,第2期
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Xu Lei,Yang Tianyu,Zhou Yiwen,Wu Meifei,Shen Jie,Cheng Jieling,Liu Qingxue,Cao Shiyang,Wang Jianqing,Zhang Lei.Bmall inhibits phenotypic transformation of hepatic stellate cells in liver fibrosis via IDH1/alpha-KG-mediated glycolysis[J].中国药理学报,2022,第2期
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Peng-xuan Ren,Wei-juan Shang,Wan-chao Yin,Huan Ge,Lin Wang,Xiang-lei Zhang,Bing-qian Li,Hong-lin Li,Ye-chun Xu,Eric H.Xu,Hua-liang Jiang,Li-li Zhu,Lei-ke Zhang,Fang Bai(School of Life Science and Technology;State Key Laboratory of Virology;CAS Key Laboratory of Receptor Research;State Key Laboratory of Bioreactor Engineering;Department of Chemistry;University of Chinese Academy of Sciences).A multi-targeting drug design strategy for identifying potent anti-SARS-CoV-2 inhibitors[J].中国药理学报(英文版),2022,第2期
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He Jiayi,Hong Quan,Chen Bixia,Cui Shaoyuan,Liu Ran,Cai Guangyan,Guo Jiao,Chen Xiangmei.Ginsenoside Rbl alleviates diabetic kidney podocyte injury by inhibiting aldose reductase activity[J].中国药理学报,2022,第2期
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Lu Qiukai,Fan Chen,Xiang Caigui,Wu Bing,Lu Huimin,Feng Chunian,Yang Xiaoqian,Li Heng,Tang Wei.Inhibition of PDE4 by apremilast attenuates skin fibrosis through directly suppressing activation of Ml and T cells[J].中国药理学报,2022,第2期
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Peng-fei Wu,Xin-lei Guan,Fang Wang,Jian-guo Chen(Department of Pharmacology;Key Laboratory of Neurological Diseases(HUST);The Key Laboratory for Drug Target Researches and Pharmacodynamic Evaluation of Hubei Province;Laboratory of Neuropsychiatric Diseases;Department of Pharmacy).N-acetylcysteine facilitates extinction of cued fear memory in rats via reestablishing basolateral amygdala glutathione homeostasis[J].中国药理学报(英文版),2022,第2期
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Zang Caixia,Wang Lu,Yang Hanyu,Shang Junmei,Liu Hui,Zhang Zihong,Ju Cheng,Yuan Fangyu,Li Fangyuan,Bao Xiuqi,Zhang Dan.HACE1 negatively regulates neuroinflammation through ubiquitylating and degrading Racl in Parkinson's disease models[J].中国药理学报,2022,第2期
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Li Wen,Liao Liping,Song Ning,Liu Yanjun,Ding Yiluan,Zhang Yuanyuan,Zhou Xiaoru,Sun Zhongya,Xiao Senhao,Wang Hongbo,Lu Jing,Zhang Naixia,Jiang Hualiang,Chen Kaixian,Liu Chuanpeng,Zheng Jie,Zhao Kehao,Luo Cheng.Natural product 1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose is a reversible inhibitor of glyceraldehyde 3-phosphate dehydrogenase[J].中国药理学报,2022,第2期
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Fei-fei Xu,Hui-min Sun,Run-ping Fang,Lu Zhang,Hui Shi,Xue Wang,Xue-li Fu,Xian-meng Li,Xu-he Shi,Yue Wu,Kai Ye,Wei-ying Zhang,Li-hong Ye(State Key Laboratory of Medicinal Chemical Biology).The modulation of PD-L1 induced by the oncogenic HBXIP for breast cancer growth[J].中国药理学报(英文版),2022,第2期
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Yu Tai,Bei Huang,Pai-pai Guo,Zhen Wang,Zheng-wei Zhou,Man-man Wang,Han-fei Sun,Yong Hu,Sheng-lin Xu,Ling-ling Zhang,Qing-tong Wang,Wei Wei(Institute of Clinical Pharmacology;Department of Pharmacy;Department of Orthopedics).TNF-α impairs EP4 signaling through the association of TRAF2-GRK2 in primary fibroblast-like synoviocytes[J].中国药理学报(英文版),2022,第2期
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Li Desheng,Xue Genlong,Yang Jiming,Li Changzhu,Zhang Ruixin,Tian Tao,Li Zheng,Shen Kewei,Guo Yang,Liu Xuening,Wang Jin,Lu Yanjie,Pan Zhenwei.Knockout of interleukin-17A diminishes ventricular arrhythmia susceptibility in diabetic mice via inhibiting NF-kappaB-mediated electrical remodeling[J].中国药理学报,2022,第2期
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Xiao-xi Hu,Ai-jun Zhang,Wen-wen Pan,Qian-ling Xin,Jing-yu Chen,Ling-ling Zhang,Yan Chang,Yu-jing Wu,Wei Wei(Institute of Clinical Pharmacology).An IgD-Fc-Ig fusion protein restrains the activation of T and B cells by inhibiting IgD-IgDR-Lck signaling in rheumatoid arthritis[J].中国药理学报(英文版),2022,第2期
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Cai-xia Zang,Lu Wang,Han-yu Yang,Jun-mei Shang,Hui Liu,Zi-hong Zhang,Cheng Ju,Fang-yu Yuan,Fang-yuan Li,Xiu-qi Bao,Dan Zhang(State Key Laboratory of Bioactive Substance and Function of Natural Medicines).HACE1 negatively regulates neuroinflammation through ubiquitylating and degrading Rac1 in Parkinson's disease models[J].中国药理学报(英文版),2022,第2期
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Susan,Wai Sum Leung,Yi Shi(Department of Pharmacology and Pharmacy;Institute of Clinical Science;Key Laboratory of Organ Transplantation).The glycolytic process in endothelial cells and its implications[J].中国药理学报(英文版),2022,第2期
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Ya-jin Lia,Rui-yuan Pan,Xiang-xi Kong,Yong Cheng,Lu Du,Zhen-chao Wang,Chao Yuan,Jin-bo Cheng,Zeng-qiang Yuan,Hai-yan Zhang(Center on Translational Neuroscience;Brain Science Center;Key Laboratory of Modern Preparation of TCM;NHC Key Laboratory of Birth Defects Research).Correction:1,2,4-Trimethoxybenzene selectively inhibits NLRP3 inflammasome activation and attenuates experimental autoimmune encephalomyelitis[J].中国药理学报(英文版),2022,第2期
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Li-wen Ren,Wan Li,Xiang-jin Zheng,Jin-yi Liu,Yi-hui Yang,Sha Li,Sen Zhang,Wei-qi Fu,Bin Xiao,Jin-hua Wang,Guan-hua Du(The State Key Laboratory of Bioactive Substance and Function of Natural Medicines;Key Laboratory of Drug Target Research and Drug Screen;Laboratory of Clinical Pharmacy).Benzimidazoles induce concurrent apoptosis and pyroptosis of human glioblastoma cells via arresting cell cycle[J].中国药理学报(英文版),2022,第1期
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Kai-long Jiang,Le-xian Tong,Tao Wang,Han-lin Wang,Xiao-bei Hu,Gao-ya Xu,Ting-ting Jin,Wei-juan Kan,Lei Xu,Jia-nan Li,Kai-xiang Zhang,Ning Song,Jie-yu Liu,Meng-meng Zhang,Wen-biao Wu,Yu-qi Xiang,An-hui Gao,Yong-zhou Hu,Yu-bo Zhou,Tao Liu,Jian-min Yang,Jia Li(National Center for Drug Screening;University of Chinese Academy of Sciences;ZJU-ENS Joint Laboratory of Medicinal Chemistry;Changhai Hospital;Shanghai Tech University;Zhongshan Institute for Drug Discovery;College of Pharmacy).Downregulation of c-Myc expression confers sensitivity to CHK1 inhibitors in hematologic malignancies[J].中国药理学报(英文版),2022,第1期
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Xin-peng Yao,Ting-ying Jiao,Yi-ming Jiang,Shi-cheng Fan,Ying-yuan Zhao,Xiao Yang,Yue Gao,Fei Li,Yan-ying Zhou,Pan-pan Chen,Min Huang,Hui-chang Bi(Guangdong Provincial Key Laboratory of New Drug Design and Evaluation;Kunming Institute of Botany;School of Pharmacy).PXR mediates mifepristone-induced hepatomegaly in mice[J].中国药理学报(英文版),2022,第1期
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Fan Yin,Pei-qing Zheng,Liu-qi Zhao,Yan-zhe Wang,Nai-jun Miao,Zhuan-li Zhou,Qian Cheng,Pan-pan Chen,Hong-yan Xie,Jing-yao Li,Jia-yun Ni,Li Zhou,Wei Zhang,Xiao-xia Wang,Jun Liu,Li-min Lu(Department of Physiology and Pathophysiology,School of Basic Medical Sciences,Fudan University,Shanghai 200032,China;Department of Nephrology,Shanghai Tong Ren Hospital,Shanghai Jiao Tong University School of Medicine,Shanghai 200336,China;Department of Physiology and Pathophysiology,School of Basic Medical Sciences,Fudan University,Shanghai 200032,China;Shanghai Kidney Development and Pediatric Kidney Disease Research Center,Shanghai 201102,China).Caspase-11 promotes NLRP3 inflammasome activation via the cleavage of pannexinl in acute kidney disease[J].中国药理学报(英文版),2022,第1期
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Ya-li Zhang,Wen-xin Zhang,Jue-qian Yan,Ye-lin Tang,Wen-jing Jia,Zheng-wei Xu,Ming-jiang Xu,Nipon Chattipakorn,Yi Wang,Jian-peng Feng,Zhi-guo Liu,Guang Liang(Chemical Biology Research Center;Key Laboratory of Molecular Pharmacology and Drug Evaluation(Yantai University);School of Pharmaceutical Sciences;Zhuji Biomedicine Institute;Cardiac Electrophysiology Research and Training Center;Wenzhou Institute).Chalcone derivatives ameliorate lipopolysaccharide-induced acute lung injury and inflammation by targeting MD2[J].中国药理学报(英文版),2022,第1期
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Li-wen Shen,Xiu-xing Jiang,Zhi-qiang Li,Jie Li,Mei Wang,Guan-fei Jia,Xin Ding,Ling Lei,Qi-hai Gong,Ning Gao(Key Laboratory of Basic Pharmacology of Ministry of Education;College of Pharmacy).Cepharanthine sensitizes human triple negative breast cancer cells to chemotherapeutic agent epirubicin via inducing cofilin oxidation-mediated mitochondrial fission and apoptosis[J].中国药理学报(英文版),2022,第1期
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Ya-lin Wang,Xiu Zhou,Dong-li Li,Ji-ming Ye(Biotechnology and Health Sciences;School of Health and Biomedical Sciences).Role of the mTOR-autophagy-ER stress pathway in high fructose-induced metabolic-associated fatty liver disease[J].中国药理学报(英文版),2022,第1期
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Yu-shan Wan,Yi You,Qian-yun Ding,Yi-xin Xu,Han Chen,Rong-rong Wang,Yu-wen Huang,Zhong Chen,Wei-wei Hu,Lei Jiang(Department of Pharmacology and Department of Pharmacy of the Second Affiliated Hospital;College of Pharmaceutical Sciences;Department of Clinical Pharmacy).Triptolide protects against white matter injury induced by chronic cerebral hypoperfusion in mice[J].中国药理学报(英文版),2022,第1期
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Mei-sa Wang,Qiu-shuang Han,Zhi-rong Jia,Chuan-sheng Chen,Chen Qiao,Qian-qian Liu,Ya-meng Zhang,Kai-wei Wang,Jie Wang,Kang Xiao,Xuan-sheng Ding(School of Basic Medicine and Clinical Pharmacy,China Pharmaceutical University,Nanjing 210009,China;Precision Medicine Laboratory,School of Basic Medicine and Clinical Pharmacy,China Pharmaceutical University,Nanjing 210009,China;School of Basic Medicine and Clinical Pharmacy,China Pharmaceutical University,Nanjing 210009,China;Department of Pharmacy,the First Affiliated Hospital of Xinjiang Medical University,Urumqi 830054,China;School of Basic Medicine and Clinical Pharmacy,China Pharmaceutical University,Nanjing 210009,China;Precision Medicine Laboratory,School of Basic Medicine and Clinical Pharmacy,China Pharmaceutical University,Nanjing 210009,China).PPARα agonist fenofibrate relieves acquired resistance to gefitinib in non-small cell lung cancer by promoting apoptosis via PPARα/AMPK/AKT/FoxOl pathway[J].中国药理学报(英文版),2022,第1期
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Ze-an Zhao,Yu Jiang,Yan-yu Chen,Ting Wu,Qun-sheng Lan,Yong-mei Li,Lu Li,Yang Yang,Cui-ting Lin,Ying Cao,Ping-zheng Zhou,Jia-yin Guo,Yuan-xin Tian,Jian-xin Pang(Guangdong Provincial Key Laboratory of Drug Screening).CDER167,a dual inhibitor of URAT1 and GLUT9,is a novel and potent uricosuric candidate for the treatment of hyperuricemia[J].中国药理学报(英文版),2022,第1期
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Chayodom Maneechote,Siripong Palee,Sasiwan Kerdphoo,Thidarat Jaiwongkam,Siriporn C.Chattipakorn,Nipon Chattipakorn(Cardiac Electrophysiology Research and Training Center;Cardiac Electrophysiology Unit;Center of Excellence in Cardiac Electrophysiology Research).Modulating mitochondrial dynamics attenuates cardiac ischemia-reperfusion injury in prediabetic rats[J].中国药理学报(英文版),2022,第1期
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Xue-qi Liu,Ling Jiang,Yuan-yuan Li,Yue-bo Huang,Xue-ru Hu,Wei Zhu,Xian Wang,Yong-gui Wu,Xiao-ming Meng,Xiang-ming Qi(Department of Nephropathy;Center for Scientific Research of Anhui Medical University;The Key Laboratory of Major Autoimmune Diseases).Wogonin protects glomerular podocytes by targeting Bcl-2-mediated autophagy and apoptosis in diabetic kidney disease[J].中国药理学报(英文版),2022,第1期
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Zhi-yun Zhu,Yan-dong Liu,Yan Gong,Wei Jin,Elena Topchiy,Subat Turdi,Yue-feng Gao,Bruce Culver,Shu-yi Wang,Wei Ge,Wen-liang Zha,Jun Ren,Zhao-hui Pei,Xing Qin(Jiangxi Provincial People’s Hospital Affiliated to Nanchang University;The Second Department of Cardiology;University of Wyoming College of Health Sciences;State Key Laboratory of Animal Nutrition;Department of General Practice;Department of Surgery;National Demonstration Center for Experimental General Medicine Education;Department of Cardiology and Shanghai Institute of Cardiovascular Diseases;Department of Cardiology).Mitochondrial aldehyde dehydrogenase(ALDH2)rescues cardiac contractile dysfunction in an APP/PS1 murine model of Alzheimer's disease via inhibition of ACSL4-dependent ferroptosis[J].中国药理学报(英文版),2022,第1期
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Dai-fei Shen,He Cheng,Bo-zhi Cai,Wen-feng Cai,Bin Wang,Qing Zhu,Yue-bin Wu,Man Liu,Run-ji Chen,Fen-fei Gao,Yan-mei Zhang,Yong-dong Niu,Gang-gang Shi(Department of Pharmacology;Qingyuan Maternal and Child Health Hospital;Laboratory of Molecular Cardiology).N-n-Butyl haloperidol iodide ameliorates liver fibrosis and hepatic stellate cell activation in mice[J].中国药理学报(英文版),2022,第1期
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Hong-yun Wang,Jun-rui Ye,Li-yuan Cui,Shi-feng Chu,Nai-hong Chen(State Key Laboratory of Bioactive Substances and Functions of Natural Medicines).Regulatory T cells in ischemic stroke[J].中国药理学报(英文版),2022,第1期
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