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冯亚美1,张强2,尹立敏1,孙隆儒1(山东大学药学院;西北农林科技大学化学与药学院).乳香中一个新的甘遂烷型三萜[J].药学学报,2022,第5期
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王冠杰1,郑海涛2,杜镇1,杨文杰1,王玥琛1,蒋海强3,4,5,田振华3,4,5(山东中医药大学药学院;平度市人民医院;山东中医药大学实验中心;山东省中医药基础研究重点实验室;山东中医药大学教育部中医药经典理论重点实验室).基于~1H NMR代谢组学及分子对接技术的异钩藤碱调控自发性高血压大鼠海马代谢研究[J].药学学报,2022,第5期
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刘春雨1,于传飞1,李欣2,付志浩1,崔永霏1,郭璐韵1,王兰1(中国食品药品检定研究院单克隆抗体产品室国家卫生健康委员会生物技术产品检定方法及其标准化重点实验室/国家药品监督管理局生物制品质量研究与评价重点实验室;广州市药品检验所).利用实验设计优化和建立抗CD38单克隆抗体ADCP生物学活性测定方法[J].药学学报,2022,第5期
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Zhu Di,Lu Yu,Gui Lin,Wang Wenjing,Hu Xi,Chen Su,Wang Yanming,Wang Yuji.Self-assembling, pH-responsive nanoflowers for inhibiting PAD4 and neutrophil extracellular trap formation and improving the tumor immune microenvironment[J].药学学报,2022,第5期
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赵梓圳,付琛,崔志鸿,李晓荣,张颖颖,张雨萍,杨晓茜,付爱玲(西南大学药学院).质子型双菲啰啉的特异性抗肿瘤活性及其机制研究[J].药学学报,2022,第5期
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Zhang Yuhong,Ding Yanqing,Li Min,Yuan Jing,Yu Youhui,Bi Xueying,Hong Huiqi,Ye Jiantao,Liu Peiqing.MicroRNA-34c-5p provokes isoprenalineinduced cardiac hypertrophy by modulating autophagy via targeting ATG4B[J].药学学报,2022,第5期
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Pan Xiaoli,Pei Junping,Wang Aoxue,Shuai Wen,Feng Lu,Bu Faqian,Zhu Yumeng,Zhang Lan,Wang Guan,Ouyang Liang.Development of small molecule extracellular signal-regulated kinases (ERKs) inhibitors for cancer therapy[J].药学学报,2022,第5期
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朱子玉,虞远智,袁月,张建军(中国医学科学院北京协和医学院药物研究所新药作用机制研究和药效评价北京市重点实验室).YZG-330通过P38 MAPK信号通路调节TRPM8离子通道发挥降温作用[J].药学学报,2022,第5期
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Liang Siping,Li Jiaying,Zou Zhengyu,Mao Miao,Ming Siqi,Lin Fan,Zhang Ziyan,Cao Can,Zhou Jinyu,Zhang Yuanqing,Li Jiaping,Wu Minhao.Tetrahedral DNA nanostructures synergize with MnO_2 to enhance antitumor immunity via promoting STING activation and M1 polarization[J].药学学报,2022,第5期
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Luo Kun,Huang Wenting,Qiao Liansheng,Zhang Xiaoling,Yan Di,Ning Zhiyu,Ma Chengmei,Dang Honglei,Wang Dong,Guo Hongyan,Xie Lan,Cheng Jing.Dendrocalamus latiflorus and its component rutin exhibit glucose-lowering activities by inhibiting hepatic glucose production via AKT activation[J].药学学报,2022,第5期
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Martin-Acosta Pedro,Meng Qianli,Klimek John,Reddy Ashok P,David Larry,Petrie Stefanie Kaech,Li Bingbing X,Xiao Xiangshu.A clickable photoaffinity probe of betulinic acid identifies tropomyosin as a target[J].药学学报,2022,第5期
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Guan Baoyi,Tong Jinlin,Hao Haiping,Yang Zhixu,Chen Keji,Xu Hao,Wang Anlu.Bile acid coordinates microbiota homeostasis and systemic immunometabolism in cardiometabolic diseases[J].药学学报,2022,第5期
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Feng Chan,Li Yongjiang,Ferdows Bijan Emiliano,Patel Dylan Neal,Ouyang Jiang,Tang Zhongmin,Kong Na,Chen Enguo,Tao Wei.Emerging vaccine nanotechnology:From defense against infection to sniping cancer[J].药学学报,2022,第5期
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Li Xuesong,Zhu Ruigong,Jiang Hong,Yin Quanwen,Gu Jiaming,Chen Jiajing,Ji Xian,Wu Xuan,Fu Haiping,Wang Hui,Tang Xin,Gao Yuanqing,Wang Bingjian,Ji Yong,Chen Hongshan.Autophagy enhanced by curcumin ameliorates inflammation in atherogenesis via the TFEB-P300-BRD4 axis[J].药学学报,2022,第5期
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Yu Weimin,Xu Gang,Chen Hui,Xiao Li,Liu Gang,Hu Pingping,Li Siqi,Kasim Vivi,Zeng Chunyu,Tong Xiaoyong.The substitution of SERCA2 redox cysteine 674 promotes pulmonary vascular remodeling by activating IRE1alpha/XBP1s pathway[J].药学学报,2022,第5期
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Yu Sifan,Li Dijie,Zhang Ning,Ni Shuaijian,Sun Meiheng,Wang Luyao,Xiao Huan,Liu Dingdong,Liu Jin,Yu Yuanyuan,Zhang Zongkang,Yeung Samuel Tin Yui,Zhang Shu,Lu Aiping,Zhang Zhenlin,Zhang Baoting,Zhang Ge.Drug discovery of sclerostin inhibitors[J].药学学报,2022,第5期
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Shen Dandan,Wang Bo,Gao Ya,Zhao Lijuan,Bi Yaping,Zhang Jinge,Wang Ning,Kang Huiqin,Pang Jingru,Liu Ying,Pang Luping,Chen Zhesheng,Zheng Yichao,Liu Hongmin.Detailed resume of RNA m~6A demethylases[J].药学学报,2022,第5期
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Zhang Youbo,Yan Tingting,Wang Tianxia,Liu Xiaoyan,Hamada Keisuke,Sun Dongxue,Sun Yizheng,Yang Yanfang,Wang Jing,Takahashi Shogo,Wang Qiong,Krausz Kristopher W,Jiang Changtao,Xie Cen,Yang Xiuwei,Gonzalez Frank J.Crosstalk between CYP2E1 and PPARalpha substrates and agonists modulate adipose browning and obesity[J].药学学报,2022,第5期
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Wang Gan,Zhang Min,Meng Ping,Long Chengbo,Luo Xiaodong,Yang Xingwei,Wang Yunfei,Zhang Zhiye,Mwangi James,Kamau Peter Muiruri,Dai Zhi,Ke Zunfu,Zhang Yi,Chen Wenlin,Zhao Xudong,Ge Fei,Lv Qiumin,Rong Mingqiang,Li Dongsheng,Jin Yang,Sheng Xia,Lai Ren.Anticarin-beta shows a promising antiosteosarcoma effect by specifically inhibiting CCT4 to impair proteostasis[J].药学学报,2022,第5期
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Luo Piao,Liu Dandan,Zhang Qian,Yang Fan,Wong Yinkwan,Xia Fei,Zhang Junzhe,Chen Jiayun,Tian Ya,Yang Chuanbin,Dai Lingyun,Shen Hanming,Wang Jigang.Celastrol induces ferroptosis in activated HSCs to ameliorate hepatic fibrosis via targeting peroxiredoxins and HO-1[J].药学学报,2022,第5期
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Chen Xiaoling,Zhang Jingliang,Wang Kewei.Inhibition of intracellular proton-sensitive Ca~(2+)-permeable TRPV3 channels protects against ischemic brain injury[J].药学学报,2022,第5期
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Xu Zhenlu,Liu Dongyun,Liu Dong,Ren Xue,Liu Haibo,Qi Guihong,Zhou Yue,Wu Chongming,Zhu Kui,Zou Zhongmei,Yuan Jing,Lin Wenhan,Guo Peng.Equisetin is an anti-obesity candidate through targeting 11beta-HSD1[J].药学学报,2022,第5期
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Liu Peihua,Jiang Ling,Kong Weimin,Xie Qiushi,Li Ping,Liu Xiaonan,Zhang Jiayi,Liu Ming,Wang Zhongjian,Zhu Liang,Yang Hanyu,Zhou Ying,Zou Jianjun,Liu Xiaodong,Liu Li.PXR activation impairs hepatic glucose metabolism partly via inhibiting the HNF4alpha-GLUT2 pathway[J].药学学报,2022,第5期
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Shi Wei,Li Wanzhen,Zhang Jianxin,Li Tiehai,Song Yakai,Zeng Yue,Dong Qian,Lin Zeng,Gong Likun,Fan Shuquan,Tang Feng,Huang Wei.One-step synthesis of site-specific antibody-drug conjugates by reprograming IgG glycoengineering with LacNAc-based substrates[J].药学学报,2022,第5期
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Liang Dong,Yu Chen,Ma Zhao,Yang Xingye,Li Zhenzhen,Dong Xuhui,Qin Xiaojun,Du Lupei,Li Minyong.Identification of anthelmintic parbendazole as a therapeutic molecule for HNSCC through connectivity map-based drug repositioning[J].药学学报,2022,第5期
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Song Nazi,Xu Hongjiao,Liu Jiahua,Zhao Qian,Chen Hui,Yan Zhibin,Yang Runling,Luo Zhiteng,Liu Qi,Ouyang Jianmei,Wu Shuohan,Luo Suijia,Ye Shuyin,Lin Runfeng,Sun Xi,Xie Junqiu,Lan Tian,Wu Zhongdao,Wang Rui,Jiang Xianxing.Design of a highly potent GLP-1R and GCGR dual-agonist for recovering hepatic fibrosis[J].药学学报,2022,第5期
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Tan Hong,Wang Huali,Ma Jinhu,Deng Hui,He Qinghua,Chen Qiang,Zhang Qinglian.Identification of human LDHC4 as a potential target for anticancer drug discovery[J].药学学报,2022,第5期
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Li Qiuyi,Chen Cheng,Kong Jinxia,Li Lian,Li Junlin,Huang Yuan.Stimuli-responsive nano vehicle enhances cancer immunotherapy by coordinating mitochondriatargeted immunogenic cell death and PD-L1 blockade[J].药学学报,2022,第5期
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Gao Wei,Hu Hongxiang,Dai Lipeng,He Miao,Yuan Hebao,Zhang Huixia,Liao Jinhui,Wen Bo,Li Yan,Palmisano Maria,Traore Mohamed Dit Mady,Zhou Simon,Sun Duxin.Structure-tissue exposure/selectivity relationship (STR) correlates with clinical efficacy/safety[J].药学学报,2022,第5期
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Fan Wufa,Peng Haixia,Yu Zhou,Wang Luting,He Haisheng,Ma Yuhua,Qi Jianping,Lu Yi,Wu Wei.The long-circulating effect of pegylated nanoparticles revisited via simultaneous monitoring of both the drug payloads and nanocarriers[J].药学学报,2022,第5期
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