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Shiqiao Peng1,Xiaoying Zhang1,Lili Yu2,Yanhong Xu3,Yang Zhou4,Shengnan Qian1,Xinyu Cao1,Xiaotong Ye4,Jiajun Yang3,Weiping Jia1,Jianping Ye1,5,6(Shanghai Diabetes Institute,Shanghai Jiao Tong University Affiliated Sixth People's Hospital;Department of Immunology,School of Basic Medical Sciences,Xinxiang Medical University;Neurology Department,Shanghai Jiao Tong University Affiliated Sixth People's Hospital;National Demonstration Center for Experimental Fisheries Science Education,College of Fisheries and Life Science,Shanghai Ocean University;Metabolic Disease Research Center,Zhengzhou University Affiliated Zhengzhou Central Hospital;Center for Advanced Medicine,College of Medicine,Zhengzhou University).NF-κB regulates brown adipocyte function through suppression of ANT2[J].Acta Pharmaceutica Sinica B,2022,第3期
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Xiaomeng Gao1,Jieqiong You1,Yanling Gong1,Meng Yuan1,2,Haiying Zhu1,Liang Fang3,Hong Zhu1,4,Meidan Ying1,4,Qiaojun He1,2,4,Bo Yang1,2,Ji Cao1,2,4(Institute of Pharmacology and Toxicology,Zhejiang Province Key Laboratory of Anti-Cancer Drug Research,College of Pharmaceutical Sciences,Zhejiang University;The Innovation Institute for Artificial Intelligence in Medicine,Zhejiang University;Department of Biology,Southern University of Science and Technology;Cancer Center of Zhejiang University).WSB1 regulates c-Myc expression through β-catenin signaling and forms a feedforward circuit[J].Acta Pharmaceutica Sinica B,2022,第3期
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Bo Zhuang1,2,Ting Chen1,Yueqi Huang1,Zhimei Xiao1,Yiguang Jin1(Department of Pharmaceutical Sciences,Beijing Institute of Radiation Medicine;Department of Chemical Defense,Institute of NBC Defense).Chemo-photothermal immunotherapy for eradication of orthotopic tumors and inhibition of metastasis by intratumoral injection of polydopamine versatile hydrogels[J].Acta Pharmaceutica Sinica B,2022,第3期
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Jingyi Li1,2,Yaqi Zhang2,3,Miaorong Yu2,Aohua Wang2,3,Yu Qiu2,3,Weiwei Fan2,Lars Hovgaard4,Mingshi Yang5,Yiming Li1,Rui Wang1,Xiuying Li6,Yong Gan2,3,7(School of Pharmacy,Shanghai University of Traditional Chinese Medicine;State Key Laboratory of Drug Research,Shanghai Institute of Materia Medica,Chinese Academy of Sciences;University of Chinese Academy of Sciences;Oral Formulation Development;Department of Pharmacy,Faculty of Health and Medical Sciences,University of Copenhagen;University of Texas at Dallas;NMPA Key Laboratory for Quality Research and Evaluation of Pharmaceutical Excipients,National Institutes for Food and Drug Control).The upregulated intestinal folate transporters direct the uptake of ligand-modified nanoparticles for enhanced oral insulin delivery[J].Acta Pharmaceutica Sinica B,2022,第3期
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Han Xiao1,2,Rui Zhang1,Xiaobo Fan1,Xinglu Jiang1,Mingyuan Zou1,Xuejiao Yan3,Haiping Hao4,Guoqiu Wu5,6(Medical School,Southeast University;Department of Clinical Laboratory,the Fifth Affiliated Hospital of Sun Yat-sen University;Department of Cardiology,the Affiliated Changzhou No.2 People's Hospital of Nanjing Medical University;State Key Laboratory of Natural Medicines,Key Lab of Drug Metabolism and Pharmacokinetics,China Pharmaceutical University;Center of Clinical Laboratory Medicine,Zhongda Hospital,Southeast University;Jiangsu Provincial Key Laboratory of Critical Care Medicine,Southeast University).Super-sensitive bifunctional nanoprobe:Self-assembly of peptide-driven nanoparticles demonstrating tumor fluorescence imaging and therapy[J].Acta Pharmaceutica Sinica B,2022,第3期
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Wenhui Tao1,Dongyang Zhao1,Guanting Li1,Lingxiao Li1,Songhao Li1,Hao Ye1,Chutong Tian1,Yutong Lu1,Shuying Li2,Yinghua Sun3,Zhonggui He1,Jin Sun1(Department of Pharmaceutics,Wuya College of Innovation,Shenyang Pharmaceutical University;Department of Pharmaceutical and Engineering,College of Pharmaceutical and Engineering,Shenyang Pharmaceutical University;Department of Pharmaceutics,College of Pharmacy,Shenyang Pharmaceutical University).Artificial tumor microenvironment regulated by first hemorrhage for enhanced tumor targeting and then occlusion for synergistic bioactivation of hypoxia-sensitive platesomes[J].Acta Pharmaceutica Sinica B,2022,第3期
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Canhao Wu1,2,Qin Xu1,Huiyuan Wang2,Bin Tu2,3,Jiaxin Zeng1,2,Pengfei Zhao2,4,Mingjie Shi2,Hong Qiu2,Yongzhuo Huang2,3,5,6(Artemisinin Research Center,First Clinical School,Guangzhou University of Chinese Medicine;State Key Laboratory of Drug Research,Shanghai Institute of Materia Medic1,Chinese Academy of Sciences;Zhongshan Institute for Drug Discovery,SIMM,CAS;Center of Clinical Pharmacology,The Second Affiliated Hospital of Zhejiang University,School of Medicine;NMPA Key Laboratory for Quality Research and Evaluation of Pharmaceutical Excipients;Taizhou University,School of Advanced Study,Institute of Natural Medicine and Health Product).Neutralization of SARS-CoV-2 pseudovirus using ACE2-engineered extracellular vesicles[J].Acta Pharmaceutica Sinica B,2022,第3期
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Shuhua Shan1,Jinping Niu1,Ruopeng Yin1,Jiangying Shi1,Lizhen Zhang2,Caihong Wu1,Hanqing Li2,Zhuoyu Li1,2(Institute of Biotechnology,Key Laboratory of Chemical Biology and Molecular Engineering of National Ministry of Education,Shanxi University;School of Life Science,Shanxi University).Peroxidase from foxtail millet bran exerts anticolorectal cancer activity via targeting cellsurface GRP78 to inactivate STAT3 pathway[J].Acta Pharmaceutica Sinica B,2022,第3期
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Chenxue Mao1,2,Juan Chen1,2,Ting Zou1,2,Yuankang Zhou1,2,Junyan Liu1,2,Xi Li1,2,Xiangping Li1,Min Li3,Pinhua Pan3,Wei Zhuo1,2,Yang Gao4,Shuo Hu5,Desheng Xiao6,Lin Wu7,Zhan Wang8,Heng Xu9,Wen Yang10,Yingjie Xu10,Haihua Xiao11,Kazuhiko Hanada12,Wei Zhang1,2,Honghao Zhou1,2,Jiye Yin1,2,Zhaoqian Liu1,2(Departments of Clinical Pharmacology and Pharmacy,Hunan Key Laboratory of Pharmacogenetics,and National Clinical Research Center for Geriatric Disorders,Xiangya Hospital,Central South University;Institute of Clinical Pharmacology,Engineering Research Center of Applied Technology of Pharmacogenomics,Ministry of Education,Central South University;Department of Respiratory,Xiangya Hospital,Central South University;Department of Thoracic Surgery,Xiangya Hospital,Central South University;Department of Nuclear Medicine,Xiangya Hospital,Central South University;Department of Pathology,Xiangya Hospital,Central South University;Department of Thoracic Medicine,Hunan Cancer Hospital;Department of Medical Oncology,Lung Cancer and Gastrointestinal Unit,Hunan Cancer Hospital;State Key Laboratory of Biotherapy and Cancer Center,West China Hospital,Sichuan University and Collaborative Innovation Center of Biotherapy;Department of Molecular and Cellular Biochemistry,School of Medicine,Shanghai Jiaotong University;Beijing National Laboratory for Molecular Sciences,State Key Laboratory of Polymer Physics and Chemistry,Institute of Chemistry,Chinese Academy of Sciences;Department of Pharmacometrics and Pharmacokinetics Meiji Pharmaceutical University).Genome-wide analysis identify novel germline genetic variations in ADCY1 influencing platinum-based chemotherapy response in nonsmall cell lung cancer[J].Acta Pharmaceutica Sinica B,2022,第3期
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Fangyu Du1,Ruolin Cao1,Lu Chen1,Jianwen Sun1,Yajie Shi1,Yang Fu1,Bruce D.Hammock2,Zhonghui Zheng3,Zhongbo Liu4,Guoliang Chen1(Key Laboratory of Structure-Based Drug Design & Discovery of Ministry of Education,School of Pharmaceutical Engineering,Shenyang Pharmaceutical University;Department of Entomology and Nematology and UC Davis Comprehensive Cancer Center,University of California Davis;Shandong Xinhua Pharmaceutical Co.,Ltd.;School of Pharmacy,Shenyang Pharmaceutical University).Structure-guided discovery of potent and oral soluble epoxide hydrolase inhibitors for the treatment of neuropathic pain[J].Acta Pharmaceutica Sinica B,2022,第3期
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Ying Zhang1,Tao Wang1,Xiaojun Zhang2,Winnie Deuther-Conrad3,Hualong Fu1,Mengchao Cui1,Jinming Zhang2,Peter Brust3,4,Yiyun Huang5,Hongmei Jia1(Key Laboratory of Radiopharmaceuticals (Beijing Normal University),Ministry of Education,College of Chemistry,Beijing Normal University;Nuclear Medicine Department,Chinese PLA General Hospital;Helmholtz-Zentrum Dresden-Rossendorf,Institute of Radiopharmaceutical Cancer Research,Department of Neuroradiopharmaceuticals;The Lübeck Institute of Experimental Dermatology,University Medical Center Schleswig-Holstein;PET Center,Department of Radiology and Biomedical Imaging,Yale University School of Medicine).Discovery and development of brain-penetrant 18F-labeled radioligands for neuroimaging of the sigma-2 receptors[J].Acta Pharmaceutica Sinica B,2022,第3期
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Wei Xie1,Shuanghuan Liu2,Guanqiao Li3,Huiyan Xu1,Liyun Zhou1(Pharmcube (Beijing) Co.,Ltd.;National Clinical Research Center for Cancer/Cancer Hospital,Chinese Academy of Medical Sciences and Peking Union Medical College;Tsinghua Clinical Research Institute (TCRI),School of Medicine,Tsinghua University).The evolving treatment paradigm of lung cancer in China[J].Acta Pharmaceutica Sinica B,2022,第3期
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Peng Teng1,Jianfeng Cai2(College of Pharmaceutical Sciences,Zhejiang University;Department of Chemistry,University of South Florida).Using proteomimetics to switch angiogenic signaling[J].Acta Pharmaceutica Sinica B,2022,第3期
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Danyu Du1,Chan Liu1,Mengyao Qin1,Xiao Zhang1,Tao Xi2,Shengtao Yuan3,Haiping Hao1,4,5,Jing Xiong1(Department of Pharmacology,School of Pharmacy,China Pharmaceutical University;Research Center of Biotechnology,School of Life Science and Technology,China Pharmaceutical University;Jiangsu Key Laboratory of Drug Screening,China Pharmaceutical University;State Key Laboratory of Natural Medicines,China Pharmaceutical University;Key Laboratory of Drug Metabolism and Pharmacokinetics,China Pharmaceutical University).Metabolic dysregulation and emerging therapeutical targets for hepatocellular carcinoma[J].Acta Pharmaceutica Sinica B,2022,第2期
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Xiang Wang1,2,Xinxin Chen3,Wenqian Zhou1,2,Hongbo Men1,2,Terigen Bao1,2,Yike Sun1,2,Quanwei Wang2,Yi Tan1,4,Bradley B.Keller4,5,6,Qian Tong2,Yang Zheng2,Lu Cai1,4(Pediatric Research Institute,Department of Pediatrics,University of Louisville School of Medicine;Department of Cardiovascular Disease,the First Hospital of Jilin University;Department of Burn Surgery,First Hospital of Jilin University,Jilin University;Department of Pharmacology and Toxicology,University of Louisville School of Medicine;Pediatric Heart Research Program,Cardiovascular Innovation Institute,University of Louisville School of Medicine;Cincinnati Children's Heart Institute,Greater Louisville and Western Kentucky Practice).Ferroptosis is essential for diabetic cardiomyopathy and is prevented by sulforaphane via AMPK/NRF2 pathways[J].Acta Pharmaceutica Sinica B,2022,第2期
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Qiubing Chen1,2,Qian Li2,Yuqi Liang1,Menghang Zu1,2,Nanxi Chen1,Brandon S.B.Canup3,Liyong Luo4,Chenhui Wang5,Liang Zeng4,Bo Xiao1,2(State Key Laboratory of Silkworm Genome Biology,College of Sericulture,Textile,and Biomass Sciences,Southwest University;Chongqing Key Laboratory of Soft-Matter Material Chemistry and Function Manufacturing,School of Materials and Energy,Southwest University;Department of Chemistry,Center for Diagnostics and Therapeutics,Georgia State University;College of Food Science,Southwest University;Chongqing Key Laboratory of Natural Product Synthesis and Drug Research,School of Pharmaceutical Sciences,Chongqing University).Natural exosome-like nanovesicles from edible tea flowers suppress metastatic breast cancer via ROS generation and microbiota modulation[J].Acta Pharmaceutica Sinica B,2022,第2期
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Makhloufi Zoulikha1,Qingqing Xiao1,George Frimpong Boafo1,Marwa A.Sallam2,Zhongjian Chen3,Wei He1,3(Department of Pharmaceutics,School of Pharmacy,China Pharmaceutical University;Department of Industrial Pharmacy,Faculty of Pharmacy,Alexandria University;Shanghai Skin Disease Hospital,Tongji University School of Medicine).Pulmonary delivery of siRNA against acute lung injury/acute respiratory distress syndrome[J].Acta Pharmaceutica Sinica B,2022,第2期
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Benjamin R.Troutwine1,2,Laylan Hamid2,Colton R.Lysaker2,3,Taylor A.Strope2,3,Heather M.Wilkins1,2,3(Department of Neurology University of Kansas Medical Center;University of Kansas Alzheimer's Disease Center;Department of Biochemistry and Molecular Biology,University of Kansas Medical Center).Apolipoprotein E and Alzheimer’s disease[J].Acta Pharmaceutica Sinica B,2022,第2期
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Eugenia Trushina1,2,Sergey Trushin1,Md Fayad Hasan1(Department of Neurology,Mayo Clinic;Department of Molecular Pharmacology and Experimental Therapeutics,Mayo Clinic).Mitochondrial complex I as a therapeutic target for Alzheimer’s disease[J].Acta Pharmaceutica Sinica B,2022,第2期
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Xiaoxi Lv1,Chang Liu1,2,Shanshan Liu1,Yunxuan Li1,Wanyu Wang1,Ke Li3,Fang Hua1,Bing Cui1,Xiaowei Zhang1,Jiaojiao Yu1,Jinmei Yu1,Zhuo Wei Hu1(Immunology and Cancer Pharmacology Group,State Key Laboratory of Bioactive Substance and Function of Natural Medicines,Institute of Materia Medica,Chinese Academy of Medical Sciences & Peking Union Medical College;Drug Clinical Trial Institution,Children's Hospital,Capital Institute of Pediatrics;Institute of Medicinal Biotechnology,Chinese Academy of Medical Sciences & Peking Union Medical College).The cell cycle inhibitor P21 promotes the development of pulmonary fibrosis by suppressing lung alveolar regeneration[J].Acta Pharmaceutica Sinica B,2022,第2期
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Xumin Zhou1,Libin Zou1,Hangyu Liao2,Junqi Luo1,Taowei Yang1,Jun Wu1,Wenbin Chen1,Kaihui Wu1,Shengren Cen1,Daojun Lv3,Fangpeng Shu4,Yu Yang5,Chun Li6,Bingkun Li1,Xiangming Mao1(Department of Urology,Zhujiang Hospital,Southern Medical University;Second Department of Hepatobiliary Surgery,Zhujiang Hospital,Southern Medical University;Department of Urology,Minimally Invasive Surgery Center,the First Affiliated Hospital of Guangzhou Medical University;Department of Urology,Guangzhou Women and Children's Medical Center,Guangzhou Medical University;Department of Urology,Peking University Shenzhen Hospital;Nursing Department,Nanfang Hospital,Southern Medical University).Abrogation of Hn RNP L enhances anti-PD-1 therapy efficacy via diminishing PD-L1 and promoting CD8+ T cell-mediated ferroptosis in castration-resistant prostate cancer[J].Acta Pharmaceutica Sinica B,2022,第2期
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Hang Qi1,Yuntao Shi2,Han Wu1,Canyang Niu1,Xiaoying Sun1,3,Ke Wei Wang1,3(Department of Pharmacology,School of Pharmacy,Qingdao University;State Key Laboratory of Natural and Biomimetic Drugs,School of Pharmaceutical Sciences,Peking University;Institue of Innovative Drugs,Qingdao University).Inhibition of temperature-sensitive TRPV3 channel by two natural isochlorogenic acid isomers for alleviation of dermatitis and chronic pruritus[J].Acta Pharmaceutica Sinica B,2022,第2期
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Mallory Little1,Moumita Dutta1,Hao Li2,Adam Matson3,Xiaojian Shi4,Gabby Mascarinas1,Bruk Molla1,Kris Weigel1,Haiwei Gu4,Sridhar Mani2,Julia Yue Cui1(Department of Environmental and Occupational Health Sciences,University of Washington;Department of Medicine,Molecular Pharmacology and Genetics,Albert Einstein College of Medicine;University of Connecticut;Arizona Metabolomics Laboratory,College of Health Solutions,Arizona State University).Understanding the physiological functions of the host xenobiotic-sensing nuclear receptors PXR and CAR on the gut microbiome using genetically modified mice[J].Acta Pharmaceutica Sinica B,2022,第2期
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Kongzhen Hu1,Junqi Li2,Lijuan Wang1,Yong Huang1,3,Li Li1,Shimin Ye1,Yanjiang Han1,Shun Huang1,Hubing Wu1,Jin Su2,4,Ganghua Tang1(Department of Nuclear Medicine,Nanfang Hospital,Southern Medical University;Shenzhen International Institute for Biomedical Research;National Cancer Center/National Clinical Research Center for Cancer/Cancer Hospital & Shenzhen Hospital,Chinese Academy of Medical Sciences and Peking Union Medical College;State Key Laboratory of Respiratory Disease,National Clinical Research Center for Respiratory Disease,Guangzhou Institute of Respiratory Health,the First Affiliated Hospital of Guangzhou Medical University).Preclinical evaluation and pilot clinical study of [18F]AlF-labeled FAPI-tracer for PET imaging of cancer associated fibroblasts[J].Acta Pharmaceutica Sinica B,2022,第2期
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Steven N.Austad1,Scott Ballinger2,Thomas W.Buford3,Christy S.Carter3,Daniel L.Smith Jr4,Victor Darley-Usmar2,Jianhua Zhang2(Department of Biology,University of Alabama at Birmingham;Department of Pathology,University of Alabama at Birmingham;Department of Medicine,University of Alabama at Birmingham;Department of Nutrition Sciences,University of Alabama at Birmingham).Targeting whole body metabolism and mitochondrial bioenergetics in the drug development for Alzheimer’s disease[J].Acta Pharmaceutica Sinica B,2022,第2期
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Shenghua Gao1,Tianguang Huang1,Letian Song1,Shujing Xu1,Yusen Cheng1,Srinivasulu Cherukupalli1,Dongwei Kang1,2,Tong Zhao1,Lin Sun1,Jian Zhang1,Peng Zhan1,2,Xinyong Liu1,2(Department of Medicinal Chemistry,Key Laboratory of Chemical Biology,Ministry of Education,School of Pharmaceutical Sciences,Cheeloo College of Medicine,Shandong University;China-Belgium Collaborative Research Center for Innovative Antiviral Drugs of Shandong Province).Medicinal chemistry strategies towards the development of effective SARS-CoV-2 inhibitors[J].Acta Pharmaceutica Sinica B,2022,第2期
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Lifang Zhao,Hongyan Zhang,Xueqing Liu,Shan Xue,Dongfang Chen,Jing Zou,Handong Jiang(Department of Respiratory and Critical Care Medicine,Ren Ji Hospital,School of Medicine,Shanghai Jiao Tong University).TGR5 deficiency activates antitumor immunity in non-small cell lung cancer via restraining M2 macrophage polarization[J].Acta Pharmaceutica Sinica B,2022,第2期
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Tao Su1,Suchao Huang1,Yanmin Zhang1,Yajuan Guo1,Shuwei Zhang1,Jiaji Guan1,Mingjing Meng1,Linxin Liu1,Caiyan Wang1,Dihua Yu2,Hiu-Yee Kwan3,Zhiying Huang1,Qiuju Huang1,Elaine Lai-Han Leung4,Ming Hue5,Ying Wang1,Zhongqiu Liu1,4,Linlin Lu1,4(Joint Laboratory for Translational Cancer Research of Chinese Medicine of the Ministry of Education of the People's Republic of China,Guangzhou University of Chinese Medicine;Department of Molecular and Cellular Oncology,the University of Texas MD Anderson Cancer Center;School of Chinese Medicine,Hong Kong Baptist University;State Key Laboratory of Quality Research in Chinese Medicine/Macau Institute for Applied Research in Medicine and Health,Macau University of Science and Technology;Department of Pharmacological and Pharmaceutical Sciences,University of Houston).miR-7/TGF-β2 axis sustains acidic tumor microenvironment-induced lung cancer metastasis[J].Acta Pharmaceutica Sinica B,2022,第2期
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