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Yinrong Wu,Zichao Yang,Kui Cheng,Huichang Bi,Jianjun Chen(Guangdong Provincial Key Laboratory of New Drug Screening,NMPA Key Laboratory for Research and Evaluation of Drug Metabolism,School of Pharmaceutical Sciences,Southern Medical University).Small molecule-based immunomodulators for cancer therapy[J].Acta Pharmaceutica Sinica B,2022,第12期
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Yanyan Xu1,Jingyuan Xiong2,Xiyang Sun3,Huile Gao1(Key Laboratory of Drug-Targeting and Drug Delivery System of the Education Ministry,Sichuan Engineering Laboratory for Plant-Sourced Drug and Sichuan Research Center for Drug Precision Industrial Technology,West China School of Pharmacy,Sichuan University;Healthy Food Evaluation Research Center,West China School of Public Health and West China Fourth Hospital,Sichuan University;Hongqiao International Institute of Medicine,Tongren Hospital,School of Medicine,Shanghai Jiao Tong University).Targeted nanomedicines remodeling immunosuppressive tumor microenvironment for enhanced cancer immunotherapy[J].Acta Pharmaceutica Sinica B,2022,第12期
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Hao Ling1,Xinyu Lou1,Qiuhua Luo2,Zhonggui He1,Mengchi Sun1,Jin Sun1(Wuya College of Innovation,Shenyang Pharmaceutical University;Department of Pharmacy,The First Affiliated Hospital of China Medical University).Recent advances in bacteriophage-based therapeutics:Insight into the post-antibiotic era[J].Acta Pharmaceutica Sinica B,2022,第12期
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Xiwei Ji1,Xiangrui Meng2,Xiao Zhu3,Qingfeng He3,Yimin Cui1(Institute of Clinical Pharmacology,Peking University First Hospital;Xiyuan Hospital,China Academy of Chinese Medical Sciences;Department of Clinical Pharmacy and Pharmacy Administration,School of Pharmacy,Fudan University).Research and development of Chinese anti-COVID-19 drugs[J].Acta Pharmaceutica Sinica B,2022,第12期
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Wan Li1,2,Hongqing Cai3,4,Liwen Ren1,2,Yihui Yang1,2,Hong Yang1,2,Jinyi Liu1,2,Sha Li1,2,Yizhi Zhang1,2,Xiangjin Zheng1,2,Wei Tan1,2,5,6,Guanhua Du1,2,Jinhua Wang1,2(The State Key Laboratory of Bioactive Substance and Function of Natural Medicines;Key Laboratory of Drug Target Research and Drug Screen,Institute of Materia Medica,Chinese Academy of Medical Science and Peking Union Medical College;Department of Neurosurgery,National Cancer Center/National Clinical Research Center for Cancer/Cancer Hospital,Chinese Academy of Medical Sciences and Peking Union Medical College;State Key Laboratory of Molecular Oncology,Center for Cancer Precision Medicine,National Cancer Center/National Clinical Research Center for Cancer/Cancer Hospital,Chinese Academy of Medical Sciences and Peking Union Medical College;School of Pharmacy,Xinjiang Medical University;Xinjiang Institute of Materia Medica).Sphingosine kinase 1 promotes growth of glioblastoma by increasing inflammation mediated by the NF-κB/IL-6/STAT3 and JNK/PTX3 pathways[J].Acta Pharmaceutica Sinica B,2022,第12期
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Minmin Fan1,2,Jian Gao1,Lin Zhou1,Wenwen Xue1,Yixuan Wang1,Jingwei Chen1,Wuhao Li1,Ying Yu1,Bo Liu3,Yan Shen1,Qiang Xu1(State Key Laboratory of Pharmaceutical Biotechnology,Nanjing Drum Tower Hospital,School of Life Sciences,Nanjing University;The First Clinical Medical College,Nanjing University of Chinese Medicine,Jiangsu Collaborative Innovation Center of Traditional Chinese Medicine Prevention and Treatment of Tumor;State Key Laboratory of Biotherapy and Cancer Center,West China Hospital,Sichuan University,Collaborative Innovation Center of Biotherapy).Highly expressed SERCA2 triggers tumor cell autophagy and is a druggable vulnerability in triple-negative breast cancer[J].Acta Pharmaceutica Sinica B,2022,第12期
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Chuchu Lin1,Chenyi Huang1,Zhaoqing Shi2,Meitong Ou1,Shengjie Sun1,Mian Yu1,Ting Chen2,Yunfei Yi1,Xiaoyuan Ji1,3,Feng Lv2,Meiying Wu1,Lin Mei2(School of Pharmaceutical Sciences (Shenzhen),Shenzhen Campus of Sun Yat-sen University;Tianjin Key Laboratory of Biomedical Materials,Key Laboratory of Biomaterials and Nanotechnology for Cancer Immunotherapy,Institute of Biomedical Engineering,Chinese Academy of Medical Sciences and Peking Union Medical College;Academy of Medical Engineering and Translational Medicine,Medical College,Tianjin University).Biodegradable calcium sulfide-based nanomodulators for H2S-boosted Ca2+-involved synergistic cascade cancer therapy[J].Acta Pharmaceutica Sinica B,2022,第12期
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Nannan Wang,Yueyue Zuo,Shengjie Wu,Chenlu Huang,Linhua Zhang,Dunwan Zhu(Tianjin Key Laboratory of Biomedical Materials,Key Laboratory of Biomaterials and Nanotechnology for Cancer Immunotherapy,Institute of Biomedical Engineering,Chinese Academy of Medical Sciences & Peking Union Medical College).Spatio-temporal delivery of both intra- and extracellular toll-like receptor agonists for enhancing antigen-specific immune responses[J].Acta Pharmaceutica Sinica B,2022,第12期
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Kai Tang,Shu Wang,Wenshuo Gao,Yihui Song,Bin Yu(School of Pharmaceutical Sciences,Zhengzhou University).Harnessing the cyclization strategy for new drug discovery[J].Acta Pharmaceutica Sinica B,2022,第12期
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Dongrong Yi1,Quanjie Li1,Han Wang2,Kai Lv1,Ling Ma1,Yujia Wang1,Jing Wang1,Yongxin Zhang1,Mingliang Liu1,Xiaoyu Li1,Jianxun Qi2,Yi Shi2,3,George F.Gao2,3,Shan Cen1,4(Institute of Medicinal Biotechnology,Chinese Academy of Medical Sciences and Peking Union Medical School;CAS Key Laboratory of Pathogenic Microbiology and Immunology,Institute of Microbiology,Chinese Academy of Sciences;University of Chinese Academy of Sciences;CAMS Key Laboratory of Antiviral Drug Research,Institute of Medicinal Biotechnology,Peking Union Medical College,Chinese Academy of Medical Sciences).Repurposing of berbamine hydrochloride to inhibit Ebola virus by targeting viral glycoprotein[J].Acta Pharmaceutica Sinica B,2022,第12期
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Yuling Mao1,Xiudan Wang1,Caishun Chen1,Qinfu Zhao1,Yanfeng Liu2,Jinghai Zhang3,Siling Wang1(Department of Pharmaceutics,School of Pharmacy,Shenyang Pharmaceutical University;School of Life Science and Bio-pharmaceutics,Shenyang Pharmaceutical University;Department of Biomedical Engineering,School of Medical Devices,Shenyang Pharmaceutical University).Immune-awakening Saccharomyces-inspired nanocarrier for oral target delivery to lymph and tumors[J].Acta Pharmaceutica Sinica B,2022,第12期
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Deying Yang1,Xiang Luo1,Qinghai Lian1,Lingqiang Gao1,Chengxin Wang1,Xiaoxiao Qi1,Rong Zhang1,Zhongqiu Liu1,2,Guochao Liao1,2(Joint Laboratory for Translational Cancer Research of Chinese Medicine of the Ministry of Education of the People’s Republic of China,International Institute for Translational Chinese Medicine,Guangzhou University of Chinese Medicine;Guangdong-Hong Kong-Macau Joint Lab on Chinese Medicine and Immune Disease Research).Fully synthetic Tn-based three-component cancer vaccine using covalently linked TLR4 ligand MPLA and iNKT cell agonist KRN-7000 as built-in adjuvant effectively protects mice from tumor development[J].Acta Pharmaceutica Sinica B,2022,第12期
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Chengliang Sun1,2,Yao Cheng1,3,Xiaojia Liu4,Gefei Wang1,2,Wenjian Min1,2,Xiao Wang1,2,Kai Yuan1,2,Yi Hou1,2,Jiaxing Li1,2,Haolin Zhang1,2,Haojie Dong1,2,Liping Wang1,2,Chenguang Lou5,Yanze Sun1,2,Xinmiao Yu1,2,Hongbin Deng6,Yibei Xiao1,3,Peng Yang1,2(State Key Laboratory of Natural Medicines and Jiangsu Key Laboratory of Drug Design and Optimization,China Pharmaceutical University;Department of Medicinal Chemistry,School of Pharmacy,China Pharmaceutical University;Department of Pharmacology,School of Pharmacy,China Pharmaceutical University;Beijing Institute of Clinical Pharmacy,Beijing Friendship Hospital,Capital Medical University;Department of Physics,Chemistry and Pharmacy,University of Southern Denmark;Institute of Medicinal Biotechnology,Chinese Academy of Medical Sciences & Peking Union Medical College).Novel phthalimides regulating PD-1/PD-L1 interaction as potential immunotherapy agents[J].Acta Pharmaceutica Sinica B,2022,第12期
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Qiang Niu1,Yu Liu2,Yujing Zheng2,Ziwei Tang1,Yuna Qian2,3,Ruogu Qi4,Jianliang Shen2,3,Ping Zhao1(School of Chemistry and Chemical Engineering,Guangdong Pharmaceutical University;State Key Laboratory of Ophthalmology,Optometry and Vision Science,School of Ophthalmology and Optometry,School of Biomedical Engineering,Wenzhou Medical University;Wenzhou Institute,University of Chinese Academy of Sciences;School of Medicine & Holistic Integrative Medicine,Nanjing University of Chinese Medicine).Co-delivery of nigericin and decitabine using hexahistidine-metal nanocarriers for pyroptosis-induced immunotherapeutics[J].Acta Pharmaceutica Sinica B,2022,第12期
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Yan-Ping Wu1,2,3,4,Rong-Rong He1,2,3,4(Guangdong Engineering Research Center of Chinese Medicine & Disease Susceptibility,Jinan University;School of Traditional Chinese Medicine,Jinan University;International Cooperative Laboratory of Traditional Chinese Medicine Modernization and Innovative Drug Development of Chinese Ministry of Education (MOE),College of Pharmacy,Jinan University;Guangdong Province Key Laboratory of Pharmacodynamic Constituents of TCM and New Drugs Research,College of Pharmacy,Jinan University).Commentary:Acute psychological stress redistributed leukocytes via distinct brain circuits[J].Acta Pharmaceutica Sinica B,2022,第12期
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Yang Liu1,Ning Zhang2,Cuicui Xie3,Yale Jiang1,Yunhe Qin3,Liyun Zhou3,Yi Fan2,Lianjie Ren2,Chen Yin1,Huan Yang2,Wei Xie3,Qing Zhai4,Guanqiao Li5,Hongzhuan Chen6,Xiaoyuan Chen1,7(Tsinghua Clinical Research Institute (TCRI),School of Medicine,Tsinghua University;Center for Drug Evaluation,National Medical Products Administration;Pharmcube (Beijing) Co.,Ltd.;Department of Clinical Pharmacy,Cancer Hospital of Fudan University;Vanke School of Public Health,Tsinghua University;Shanghai Collaborative Innovation Center for Translational Medicine,Shanghai University of Traditional Chinese Medicine;Office of Clinical Trial Institute,Beijing Tsinghua Changgung Hospital).Evolution of drug regulations and regulatory innovation for anticancer drugs in China[J].Acta Pharmaceutica Sinica B,2022,第12期
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Shujing Xu,Xinyong Liu,Peng Zhan(Department of Medicinal Chemistry,Key Laboratory of Chemical Biology,Ministry of Education,School of Pharmaceutical Sciences,Shandong University).SMIP-30, a potent and selective PPM1A inhibitor with potential to treat tuberculosis[J].Acta Pharmaceutica Sinica B,2022,第12期
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Yuyu Zhu1,Zijun Ouyang2,Haojie Du3,Meijing Wang3,Jiaojiao Wang1,Haiyan Sun2,Lingdong Kong3,Qiang Xu3,Hongyue Ma1,Yang Sun3,4(College of Pharmacy,Nanjing University of Chinese Medicine;Institute of Marine Biomedicine,School of Food and Drug,Shenzhen Polytechnic;State Key Laboratory of Pharmaceutical Biotechnology,School of Life Science,Nanjing University;Jiangsu Key Laboratory of New Drug Research and Clinical Pharmacy,Xuzhou Medical University).New opportunities and challenges of natural products research:When target identification meets single-cell multiomics[J].Acta Pharmaceutica Sinica B,2022,第11期
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Shilin Chen1,2,Zheng Li3,Sanyin Zhang4,Yuxin Zhou1,2,Xiaohe Xiao5,Pengdi Cui3,Binjie Xu4,Qinghe Zhao2,Shasha Kong2,Yuntao Dai2(Institute of Herbgenomics,Chengdu University of Traditional Chinese Medicine;Institute of Chinese Materia Medica,China Academy of Chinese Medical Sciences;State Key Laboratory of Component Traditional Chinese Medicine,College of Pharmaceutical Engineering of Traditional Chinese Medicine,Haihe Laboratory of Modern Chinese Medicine,Tianjin University of Traditional Chinese Medicine;Innovative Institute of Chinese Medicine and Pharmacy,Chengdu University of Traditional Chinese Medicine;China Military Institute of Chinese Medicine,Fifth Medical Center of Chinese PLA General Hospital).Emerging biotechnology applications in natural product and synthetic pharmaceutical analyses[J].Acta Pharmaceutica Sinica B,2022,第11期
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Xiaoyou Wang1,Chong Li1,Yiguang Wang2,Huabing Chen3,Xinxin Zhang4,Cong Luo5,Wenhu Zhou6,Lili Li7,Lesheng Teng8,Haijun Yu4,Jiancheng Wang2(College of Pharmaceutical Sciences,Southwest University;Beijing Key Laboratory of Molecular Pharmaceutics and New Drug Delivery Systems,State Key Laboratory of Natural and Biomimetic Drugs,School of Pharmaceutical Sciences,Peking University;School of Radiation Medicine and Protection,Soochow University;Shanghai Institute of Materia Medica,Chinese Academy of Sciences;Department of Pharmaceutics,Wuya College of Innovation,Shenyang Pharmaceutical University;Xiangya School of Pharmaceutical Sciences,Central South University;CAS Center for Excellence in Nanoscience,CAS Key Laboratory for Biomedical Effects of Nanomaterials and Nanosafety,National Center for Nanoscience and Technology;School of Life Sciences,Jilin University).Smart drug delivery systems for precise cancer therapy[J].Acta Pharmaceutica Sinica B,2022,第11期
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Saiyang Xie1,2,Yun Xing1,2,Wenke Shi1,2,Min Zhang1,2,Mengya Chen1,2,Wenxi Fang1,2,Shiqiang Liu1,2,Tong Zhang1,2,Xiaofeng Zeng3,Si Chen3,Shasha Wang3,Wei Deng1,2,Qizhu Tang1,2(Department of Cardiology,Renmin Hospital of Wuhan University;Hubei Key Laboratory of Metabolic and Chronic Diseases;Cardiovascular Research Institute of Wuhan University).Cardiac fibroblast heat shock protein 47 aggravates cardiac fibrosis post myocardial ischemia-reperfusion injury by encouraging ubiquitin specific peptidase 10 dependent Smad4 deubiquitination[J].Acta Pharmaceutica Sinica B,2022,第11期
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Liping Liao1,2,Wenzhen Dang3,1,Tingting Lin1,2,Jinghua Yu1,Tonghai Liu1,2,Wen Li1,Senhao Xiao1,2,Lei Feng1,2,Jing Huang1,2,Rong Fu1,Jiacheng Li1,2,Liping Liu1,2,Mingchen Wang1,2,Hongru Tao1,Hualiang Jiang1,2,Kaixian Chen1,2,Xingxing Diao1,Bing Zhou1,4,Xiaoyan Shen3,Cheng Luo3,1,2,4,5(State Key Laboratory of Drug Research,Shanghai Institute of Materia Medica,Chinese Academy of Sciences;University of Chinese Academy of Sciences;Department of Pharmacology & the Key Laboratory of Smart Drug Delivery,Ministry of Education,School of Pharmacy,Fudan University;School of Pharmaceutical Science and Technology,Hangzhou Institute for Advanced Study,University of Chinese Academy of Sciences;School of Pharmaceutical Sciences,Zhejiang Chinese Medical University).A potent PGK1 antagonist reveals PGK1 regulates the production of IL-1β and IL-6[J].Acta Pharmaceutica Sinica B,2022,第11期
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Juan Pang1,2,Jia Nuo Feng2,3,Wenhua Ling1,Tianru Jin2,3,4(Department of Nutrition,School of Public Health,Sun Yat-sen Universitynstitute;Division of Advanced Diagnostics,Toronto General Hospital Research Ⅰ,University Health Network;Department of Physiology,Faculty of Medicine,University of Toronto;Banting and Best Diabetes Centre,Faculty of Medicine,University of Toronto).The anti-inflammatory feature of glucagon-like peptide-1 and its based diabetes drugs——Therapeutic potential exploration in lung injury[J].Acta Pharmaceutica Sinica B,2022,第11期
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Jie Tu,Na Liu,Yahui Huang,Wanzhen Yang,Chunquan Sheng(School of Pharmacy,Second Military Medical University).Small molecules for combating multidrug-resistant superbug Candida auris infections[J].Acta Pharmaceutica Sinica B,2022,第11期
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Yan Li1,2,Ya Chu1,3,Guangjiang Shi1,3,Xiaobin Wang1,Wanli Ye1,3,Chun Shan1,Dajia Wang1,Di Zhang3,Wei He3,Jingwei Jiang4,Shuqian Ma1,3,Yuhong Han1,3,Zhili Zhao1,Shijia Du1,Zhen Chen3,Zhiyu Li3,Yong Yang1,Chen Wang2,Xi Xu3,Hongxi Wu3(Center for New Drug Safety Evaluation and Research,State Key Laboratory of Natural Medicines,China Pharmaceutical University;School of Life Science and Technology,China Pharmaceutical University;School of Pharmacy,China Pharmaceutical University;Jiangsu Key Lab of Drug Screening,China Pharmaceutical University).A novel inhibitor of ARfl and ARv7 induces protein degradation to overcome enzalutamide resistance in advanced prostate cancer[J].Acta Pharmaceutica Sinica B,2022,第11期
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Beifen Zhong1,Jun Wan1,Changhui Shang1,Jiajia Wen2,Yujia Wang2,Jian Bai1,Shan Cen2,Youcai Hu1(State Key Laboratory of Bioactive Substance and Function of Natural Medicines,Institute of Materia Medica,Chinese Academy of Medical Sciences & Peking Union Medical College;Institute of Medicinal Biotechnology,Chinese Academy of Medical Sciences & Peking Union Medical College).Biosynthesis of rumbrins and inspiration for discovery of HIV inhibitors[J].Acta Pharmaceutica Sinica B,2022,第11期
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Zaigang Zhou1,2,Jiashe Chen3,Yu Liu1,Chunjuan Zheng4,Wenjuan Luo4,Lele Chen3,Shen Zhou3,Zhiming Li3,Jianliang Shen1,2,5(State Key Laboratory of Ophthalmology,Optometry and Vision Science,School of Ophthalmology and Optometry,School of Biomedical Engineering,Wenzhou Medical University;Wenzhou Institute,University of Chinese Academy of Sciences;Department of the First Affiliated Hospital of Wenzhou Medical University;School & Hospital of Stomatology,Wenzhou Medical University;Oujiang Laboratory(Zhejiang Lab for Regenerative Medicine,Vision and Brain Health)).Cascade two-stage tumor re-oxygenation and immune re-sensitization mediated by self-assembled albumin-sorafenib nanoparticles for enhanced photodynamic immunotherapy[J].Acta Pharmaceutica Sinica B,2022,第11期
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Zekun Li1,Yongchun Pan2,Shiyu Du1,Yayao Li1,Chao Chen1,Hongxiu Song1,Yueyao Wu1,Xiaowei Luan2,Qin Xu2,Xiaoxiang Guan3,Yujun Song2,Xin Han1(Jiangsu Key Laboratory for Pharmacology and Safety Evaluation of Chinese Materia Medica,School of Medicine& Holistic Integrative Medicine,Jiangsu Joint International Research Laboratory of Chinese Medicine and Regenerative Medicine,Nanjing University of Chinese Medicine;College of Engineering and Applied Sciences,Jiangsu Key Laboratory of Artificial Functional Materials,State Key Laboratory of Analytical Chemistry for Life Science,Nanjing University;Department of Oncology,The First Affiliated Hospital of Nanjing Medical University).Tumor-microenvironment activated duplex genome-editing nanoprodrug for sensitized near-infrared titania phototherapy[J].Acta Pharmaceutica Sinica B,2022,第11期
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Chunying Liu1,Shuangrong Ruan2,Ying He1,Xuejing Li1,Yuefei Zhu1,3,Honglan Wang4,Hanwei Huang1,Zhiqing Pang1(School of Pharmacy,Fudan University,Key Laboratory of Smart Drug Delivery,Ministry of Education;The Institute for Biomedical Engineering & Nano Science,Tongji University School of Medicine;Department of Biomedical Engineering,Columbia University;Institute of Hematology,Union Hospital,Tongji Medical College,Huazhong University of Science & Technology).Broad-spectrum and powerful neutralization of bacterial toxins by erythroliposomes with the help of macrophage uptake and degradation[J].Acta Pharmaceutica Sinica B,2022,第11期
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